PDE inhibitor

PDE inhibitor
inhibiteur de la phosphodiestérase

English-French medical dictionary. 2015.

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  • PDE-5 inhibitor — ▪ category of drugs in full  phosphodiesterase 5 inhibitor        category of drugs that relieve erectile dysfunction ( impotence) in men. Two common commercially produced PDE 5 inhibitors are sildenafil (sold as Viagra) and vardenafil (Levitra) …   Universalium

  • PDE-5-Inhibitor — Phosphodiesterase 5 Hemmer (auch Phosphodiesterase V Hemmer, PDE 5 Hemmer) sind Substanzen, die das cGMP abbauende Enzym Phosphodiesterase V hemmen und somit die Konzentration von intrazellulärem cGMP (zyklisches Guanosinmonophosphat) erhöhen.… …   Deutsch Wikipedia

  • PDE-V-Inhibitor — Phosphodiesterase 5 Hemmer (auch Phosphodiesterase V Hemmer, PDE 5 Hemmer) sind Substanzen, die das cGMP abbauende Enzym Phosphodiesterase V hemmen und somit die Konzentration von intrazellulärem cGMP (zyklisches Guanosinmonophosphat) erhöhen.… …   Deutsch Wikipedia

  • PDE-V-Hemmer — Phosphodiesterase 5 Hemmer (auch Phosphodiesterase V Hemmer, PDE 5 Hemmer) sind Substanzen, die das cGMP abbauende Enzym Phosphodiesterase V hemmen und somit die Konzentration von intrazellulärem cGMP (zyklisches Guanosinmonophosphat) erhöhen.… …   Deutsch Wikipedia

  • PDE3 inhibitor — Milrinone, one of the first PDE3 inhibitors used clinically A PDE3 inhibitor is a drug which inhibits the action of the phosphodiesterase enzyme PDE3. They are used for the therapy of acute heart failure and cardiogenic shock. Approved PDE3… …   Wikipedia

  • Phosphodiesterase inhibitor — A phosphodiesterase inhibitor is a drug that blocks one or more of the five subtypes of the enzyme phosphodiesterase (PDE), therefore preventing the inactivation of the intracellular second messengers cyclic adenosine monophosphate (cAMP) and… …   Wikipedia

  • PDE4 inhibitor — Piclamilast, a common PDE4 inhibitor A phosphodiesterase type 4 inhibitor, commonly referred to as a PDE4 inhibitor, is a drug used to block the degradative action of phosphodiesterase 4 (PDE4) on cyclic adenosine monophosphate (cAMP). It is a… …   Wikipedia

  • PDE5 inhibitor — Sildenafil (Viagra), the prototypical PDE5 inhibitor A phosphodiesterase type 5 inhibitor, often shortened to PDE5 inhibitor, is a drug used to block the degradative action of phosphodiesterase type 5 on cyclic GMP in the smooth muscle cells… …   Wikipedia

  • Phosphodiesterase-5-Inhibitor — Phosphodiesterase 5 Hemmer (auch Phosphodiesterase V Hemmer, PDE 5 Hemmer) sind Substanzen, die das cGMP abbauende Enzym Phosphodiesterase V hemmen und somit die Konzentration von intrazellulärem cGMP (zyklisches Guanosinmonophosphat) erhöhen.… …   Deutsch Wikipedia

  • Phosphodiesterase-V-Inhibitor — Phosphodiesterase 5 Hemmer (auch Phosphodiesterase V Hemmer, PDE 5 Hemmer) sind Substanzen, die das cGMP abbauende Enzym Phosphodiesterase V hemmen und somit die Konzentration von intrazellulärem cGMP (zyklisches Guanosinmonophosphat) erhöhen.… …   Deutsch Wikipedia

  • Ibudilast — Drugbox IUPAC name = 2 methyl 1 (2 propan 2 ylpyrazolo [1,5 a] pyridin 3 yl)propan 1 one CAS number = 50847 11 5 ATC prefix = ATC suffix = PubChem = 3671 DrugBank = C=14|H=18|N=2|O=1 molecular weight = 230.31 g/mol bioavailability = protein bound …   Wikipedia

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